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8 times the recommended single dose with a moderate cyp3a4 inhibitor, diltiazem, increased the aprepitant auc 2-fold with a concomitant 1.
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there were seven reports with a fatal outcome; although the amount of diltiazem ingested was unknown, multiple drug ingestions were confirmed in six of the seven reports.
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there have been 29 reports of diltiazem overdose in doses ranging from less than 1 gm to 10.
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